SCHEMBL7367864

SCHEMBL7367864

COc1ccc(O)c(CCC(=O)OC(C)(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.55
MTNR1A P48039 1/20 0.52
MTNR1B P49286 1/20 0.52
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
PKM P14618 1/20 0.47
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
HSD17B10 Q99714 1/20 0.43
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21437958 0.85 MTNR1A (0.51) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL7373176 0.83 CYP3A4 (0.48) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL31587683 0.83 CA12 (0.39) POLBMTNR1AMTNR1BCA1
SCHEMBL7368806 0.82 POLB (0.79) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL7373180 0.81 POLB (0.44) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL8413349 0.81 PRKCI (0.44) POLBHSD17B10
SCHEMBL6036442 0.81 POLB (0.56) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL7453167 0.80 POLB (0.40) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL7453174 0.80 POLB (0.40) POLBMTNR1AMTNR1BNPC1RAB9A
SCHEMBL7453171 0.80 POLB (0.43) POLBMTNR1AMTNR1BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000031-A4 VITRONECTIN RECEPTOR ANTAGONIST SMITHKLINE BEECHAM CORP (US) 2001-08-16 EP disclosed
US-6239138-B1 TREATMENT OF INFLAMMATION, CANCER, CARDIOVASCULAR DISORDERS, SUCH AS ATHEROSCLEROSIS AND RESTENOSIS, OSTEOPOROSIS, BENZOCYCLOHEPTENYL IN WHICH A NITROGEN-CONTAINING SUBSTITUENT IS PRESENT ON THE AROMATIC SIX-MEMBERED RING AND AN ALIPHATIC SMITHKLINE BEECHAM CORPORATION 2001-05-29 US disclosed
EP-1000031-A1 VITRONECTIN RECEPTOR ANTAGONIST SmithKline Beecham Corporation (US) 2000-05-17 EP disclosed
WO-1999005107-A1 VITRONECTIN RECEPTOR ANTAGONIST SMITHKLINE BEECHAM CORPORATION (US) 1999-02-04 WO disclosed