SCHEMBL7369068

SCHEMBL7369068

O=c1cccc(-c2ccc(Br)cc2)[nH]1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.67
MAP2K1 Q02750 1/20 0.59
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
MMP1 P03956 1/20 0.41
ALDH1A1 P00352 4/20 0.41
TSHR P16473 1/20 0.41
IDO1 P14902 1/20 0.40
MAPK1 P28482 1/20 0.39
BRS3 P32247 1/20 0.38
TNKS O95271 3/20 0.38
TNKS2 Q9H2K2 3/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1384813 0.80 NOTUM (1.00) NOTUMMAP2K1GAAMAPTALDH1A1
SCHEMBL7368040 0.80 NOTUM (0.62) NOTUMMAP2K1GAAMMP1ALDH1A1
SCHEMBL5674033 0.79 NOTUM (0.67) NOTUMMAP2K1MEN1KMT2AGAA
SCHEMBL8535240 0.77 NOTUM (0.68) NOTUMMAP2K1MMP1ALDH1A1CYP1A1
SCHEMBL17488164 0.76 NOTUM (0.62) NOTUMMAP2K1ALDH1A1BRS3GCK
SCHEMBL11226843 0.75 NOTUM (0.67) NOTUMMAP2K1MAPTMAPK1CDK1
Hydrochloric Acid SCHEMBL31700388 0.75 NOTUM (0.60) NOTUMMAP2K1GAAMAPTBRS3
SCHEMBL26033405 0.75 NOTUM (0.60) NOTUMMAP2K1MEN1KMT2AMAPT
SCHEMBL26953393 0.75 NOTUM (0.55) NOTUMMAP2K1BRS3CA12CA9
SCHEMBL3072721 0.75 NOTUM (0.66) NOTUMMAP2K1KMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613467-A1 2-PYRIDINOL DERIVATIVES AND THEIR USE AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1994-09-07 EP disclosed
WO-1993010093-A1 2-PYRIDINOL DERIVATIVES AND THEIR USE AS MEDICAMENTS SMITHKLINE BEECHAM PLC (GB) 1993-05-27 WO disclosed