SCHEMBL7369390

SCHEMBL7369390

CCOC(=O)C=Cc1ccc(O)c(Cl)c1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TTR P02766 4/20 0.76
DPP4 P27487 1/20 0.76
MAOB P27338 1/20 0.68
CYP3A4 P08684 1/20 0.63
CA12 O43570 1/20 0.63
CA1 P00915 1/20 0.63
CA2 P00918 1/20 0.63
CA7 P43166 1/20 0.63
CA9 Q16790 1/20 0.63
CA14 Q9ULX7 1/20 0.63
APP P05067 9/20 0.59
BACE1 P56817 1/20 0.57
FDPS P14324 1/20 0.54
AKR1B10 O60218 1/20 0.50
AKR1B1 P15121 1/20 0.50
ESR1 P03372 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2388953 1.00 TTR (0.76) TTRDPP4MAOBCYP3A4CA12
SCHEMBL2259487 0.88 TTR (0.76) TTRDPP4MAOBCYP3A4CA12
SCHEMBL2259482 0.88 TTR (0.76) TTRDPP4MAOBCYP3A4CA12
SCHEMBL1713415 0.88 TTR (0.66) TTRDPP4MAOBCYP3A4CA12
SCHEMBL1713417 0.88 TTR (0.66) TTRDPP4MAOBCYP3A4CA12
SCHEMBL9862625 0.87 TTR (0.64) TTRDPP4MAOBCYP3A4CA12
SCHEMBL9862626 0.87 TTR (0.64) TTRDPP4MAOBCYP3A4CA12
Ethyl Caffeate SCHEMBL782033 0.86 TTR (1.00) TTRDPP4MAOBCYP3A4CA12
Ethyl Caffeate SCHEMBL22196845 0.86 TTR (1.00) TTRDPP4MAOBCYP3A4CA12
Ethyl Caffeate SCHEMBL782032 0.86 TTR (1.00) TTRDPP4MAOBCYP3A4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5137889-A Hypotensive agents; coronary vasodilators; calcium antagonists; antiinflammatory agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-08-11 US disclosed
US-5034395-A Hypotensive agents, carboxylated dihydropyridines OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-07-23 US disclosed
US-4795814-A CORONARY VASODILATORS, HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANTITUMOR AGENTTS, ENZYME INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-01-03 US disclosed
EP-0145434-A2 Novel dihydropyridine derivatives and process for preparing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1985-06-19 EP disclosed