SCHEMBL7370980

SCHEMBL7370980

CCOC(=O)[C@H](Cc1ccccc1)NC(=O)CNc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.56
TACR1 P25103 1/20 0.55
ALDH1A1 P00352 4/20 0.50
POLB P06746 2/20 0.50
THRB P10828 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MMP8 P22894 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
EGFR P00533 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365183 0.88 TACR1 (0.60) TACR1ALDH1A1POLBTHRBCYP2C9
SCHEMBL9487298 0.85 TP53 (0.61) TP53TACR1ALDH1A1POLBMMP8
SCHEMBL9487303 0.85 TP53 (0.61) TP53TACR1ALDH1A1POLBMMP8
SCHEMBL9146870 0.83 TP53 (0.60) TP53TACR1ALDH1A1POLBTHRB
SCHEMBL9385733 0.83 TP53 (0.60) TP53TACR1ALDH1A1POLBTHRB
SCHEMBL11559927 0.83 TP53 (0.60) TP53TACR1ALDH1A1POLBMMP8
SCHEMBL9146866 0.83 TP53 (0.60) TP53TACR1ALDH1A1POLBTHRB
SCHEMBL9385728 0.83 TP53 (0.60) TP53TACR1ALDH1A1POLBTHRB
SCHEMBL7365767 0.83 MME (0.55)
SCHEMBL9488182 0.82 TP53 (0.59) TP53TACR1ALDH1A1POLBMMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001973-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006433-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed