SCHEMBL7372992

SCHEMBL7372992

CCOC(=O)C1=C(C(OCC)OCC)NC(C)=C(C(=O)O)C1c1ccccc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.42
CYP2C9 P11712 4/20 0.42
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C19 P33261 3/20 0.42
ADORA3 P0DMS8 2/20 0.42
KDM4E B2RXH2 4/20 0.41
HSD17B10 Q99714 3/20 0.41
CASP1 P29466 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HIF1A Q16665 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
GAA P10253 2/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381384 0.85 ADORA3 (0.46) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL7380766 0.84 ADORA3 (0.46) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7158453 0.83 ADORA3 (0.55) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7374894 0.82 NR1I2 (0.44) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7383456 0.82 CACNA1C (0.46) CACNA1C
SCHEMBL7380754 0.82 CACNA1C (0.55) CACNA1C
SCHEMBL7384393 0.82 CACNA1C (0.43) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7379022 0.79 KDM4E (0.57) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL10642720 0.79 KDM4E (0.47) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL11693531 0.79 CYP2C9 (0.51) CACNA1CCYP2C9CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4525478-A Certain 4-aryl-1,4-dihydro-3,5-pyridinedicarboxylates having vasodilating and anti-hypertensive properties FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1985-06-25 US disclosed
US-4393070-A HYPOTENSIVE, VASODILATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-07-12 US disclosed
US-4370334-A VASODILATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-01-25 US disclosed
US-4338322-A 1,4-Dihydropyridine derivatives, pharmaceutical compositions containing same and methods of effecting vasodilation using same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1982-07-06 US disclosed
US-4307103-A TREATMENT OF HYPERTENSION AND CARDIOVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-12-22 US disclosed
US-4284634-A HYPOTENSIVE VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-08-18 US disclosed