SCHEMBL7373407

SCHEMBL7373407

Cc1ncccc1OC[C@H]1CCN1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.81
CHRNA4 P43681 3/20 0.81
CHRNA3 P32297 4/20 0.58
CHRNB4 P30926 3/20 0.58
CHRNB1 P11230 2/20 0.56
CHRNB3 Q05901 1/20 0.56
CHRNA7 P36544 2/20 0.55
CHRNA1 P02708 1/20 0.55
CHRNG P07510 1/20 0.55
CHRND Q07001 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL905231 1.00 CHRNB2 (0.81) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Hydrochloric Acid SCHEMBL7450656 0.98 CHRNB2 (0.78) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Hydrochloric Acid SCHEMBL7415362 0.98 CHRNB2 (0.78) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL7367252 0.89 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL194037 0.89 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL1538473 0.89 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL29378392 0.89 CHRNB2 (1.00) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL29711154 0.88 CHRNB2 (0.97) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL7838537 0.88 CHRNB2 (0.97) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
Pozanicline SCHEMBL5139644 0.88 CHRNB2 (0.97) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663912-B1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LAB (US) 2001-12-12 EP claimed
US-5948793-A 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release ABBOTT LABORATORIES (US) 1999-09-07 US claimed
EP-0663912-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1995-07-26 EP claimed
EP-0663912-A4 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION. ABBOTT LAB (US) 1995-02-17 EP claimed
WO-1994008992-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1994-04-28 WO claimed
EP-0663912-B1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LAB (US) 2001-12-12 EP disclosed
US-5948793-A 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release ABBOTT LABORATORIES (US) 1999-09-07 US disclosed
EP-0663912-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1995-07-26 EP disclosed
EP-0663912-A4 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION. ABBOTT LAB (US) 1995-02-17 EP disclosed
WO-1994008992-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1994-04-28 WO disclosed