SCHEMBL7373771

SCHEMBL7373771

O=C(O)CNC(=O)c1cc(NC2=NCCN2)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.47
ITGAV P06756 13/20 0.47
ITGB6 P18564 11/20 0.47
ITGB1 P05556 6/20 0.47
ITGA5 P08648 6/20 0.47
ITGB5 P18084 6/20 0.47
ITGB8 P26012 6/20 0.47
ITGA8 P53708 6/20 0.47
PTGIR P43119 1/20 0.44
ADRA2A P08913 2/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
WDR5 P61964 1/20 0.42
EGLN1 Q9GZT9 1/20 0.40
RHOC P08134 1/20 0.40
RHOA P61586 1/20 0.40
SYK P43405 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7844560 0.99 ITGB3 (0.47) ITGB3ITGAVITGB6ITGB1ITGA5
Hydrochloric Acid SCHEMBL6224028 0.79 ITGB3 (0.58) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL29448189 0.79 ITGB3 (0.75) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7501057 0.78 ITGB3 (0.52) ITGB3ITGAVITGB1ITGB5WDR5
SCHEMBL7501047 0.78 ITGB3 (0.52) ITGB3ITGAVITGB1ITGB5WDR5
SCHEMBL19265544 0.78 ITGB3 (0.63) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL8443562 0.77 ITGB3 (0.51) ITGB3ITGAVITGB1ITGB5
SCHEMBL615919 0.75 TACR1 (0.59) EGLN1RHOCRHOA
SCHEMBL6778283 0.75 ITGB3 (0.64) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL8542414 0.74 PTGIR (0.39) ITGB3ITGAVITGB6ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed