SCHEMBL7374841

SCHEMBL7374841

O=C[C@H](Cc1ccccc1)NC(=O)c1ccc(NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
CAPN1 P07384 5/20 0.53
TDP1 Q9NUW8 1/20 0.52
HDAC1 Q13547 3/20 0.51
CASP3 P42574 1/20 0.47
HDAC8 Q9BY41 2/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7791366 1.00 MEN1 (0.53) MEN1KMT2ACAPN1TDP1HDAC1
SCHEMBL7787808 0.88 ALDH1A1 (0.56) MEN1KMT2ACAPN1HDAC1HDAC8
SCHEMBL7787807 0.88 ALDH1A1 (0.56) MEN1KMT2ACAPN1HDAC1HDAC8
SCHEMBL7378076 0.87 CAPN1 (0.53) MEN1KMT2ACAPN1HDAC8HDAC2
SCHEMBL7782239 0.87 CAPN1 (0.53) MEN1KMT2ACAPN1HDAC8HDAC2
SCHEMBL7786963 0.82 CAPN1 (0.50) CAPN1HDAC1ALDH1A1
SCHEMBL7786967 0.82 CAPN1 (0.50) CAPN1HDAC1ALDH1A1
SCHEMBL7782130 0.82 MAPK1 (0.58) MEN1KMT2ATDP1HDAC1HDAC8
SCHEMBL7380786 0.82 MAPK1 (0.58) MEN1KMT2ATDP1HDAC1HDAC8
SCHEMBL40781 0.82 CAPN1 (0.74) CAPN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
EP-0944584-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998023581-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-04 WO disclosed