SCHEMBL7375302

SCHEMBL7375302

CC(C)(C)OC(=O)Nc1ccc(CN2CCNCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.52
PTGDR2 Q9Y5Y4 1/20 0.49
CYP17A1 P05093 1/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
SLC2A1 P11166 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
POLB P06746 1/20 0.45
CD274 Q9NZQ7 1/20 0.45
MAPT P10636 1/20 0.45
CXCR4 P61073 2/20 0.44
MEN1 O00255 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
ADRA2C P18825 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28802622 0.88 KDM4E (0.63) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL1604864 0.87 KDM4E (0.66) DRD2CYP17A1KDM4EALDH1A1POLB
SCHEMBL22571323 0.85 CD274 (0.61) ALDH1A1RAB9ANPC1POLBCD274
SCHEMBL7372715 0.82 DRD2 (0.53) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL22872079 0.81 DRD2 (0.49) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL15858103 0.81 CD274 (0.43) DRD2ALDH1A1RAB9ANPC1TP53
SCHEMBL15853663 0.81 CYP17A1 (0.74) DRD2PTGDR2CYP17A1KDM4EALDH1A1
SCHEMBL31047972 0.80 CXCR4 (0.48) KDM4ECXCR4MEN1CHRM2CHRM1
SCHEMBL6503210 0.80 MAPT (0.50) KDM4EALDH1A1RAB9ANPC1TP53
SCHEMBL28698604 0.80 DRD2 (0.53) DRD2PTGDR2CYP17A1ALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929074-A VSODILATOR, ANTIALLERGIC AND ANTIPLATELET AGENTS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-27 US disclosed
EP-0706517-B1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL IND LTD (JP) 1998-10-21 EP disclosed
EP-0706517-A1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1996-04-17 EP disclosed
WO-1995001343-A1 PYRIDAZINONE DERIVATIVES WITH PHARMACEUTICAL ACTIVITY NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1995-01-12 WO disclosed