SCHEMBL7375827

SCHEMBL7375827

O=c1ccccn1C1=CC2(CCCCC2)Oc2ncccc21

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
CTSL P07711 1/20 0.30
PTPRC P08575 1/20 0.30
CTSS P25774 1/20 0.30
PTPN13 Q12923 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374473 0.99 PTPRC (0.31) CTSLPTPRCCTSSPTPN13
SCHEMBL7372034 0.84 EPHX2 (0.32) ALDH1A1
SCHEMBL7368502 0.82 EPHX2 (0.32)
SCHEMBL7299641 0.81 HRH4 (0.33)
SCHEMBL7374320 0.78 CA12 (0.37) ALDH1A1
SCHEMBL7371741 0.78 HASPIN (0.38)
SCHEMBL7371009 0.77 CA12 (0.38) ALDH1A1
SCHEMBL7373810 0.77 CA12 (0.38)
SCHEMBL8084291 0.71 OPRD1 (0.39)
SCHEMBL8090132 0.71 OPRD1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308792-B1 AZACHROMANE DERIVATIVES MERCK PATENT GmbH (DE) 1993-07-28 EP disclosed
US-4931454-A Azachroman derivatives with effects on the cardiovascular system MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-06-05 US disclosed