SCHEMBL7377883

SCHEMBL7377883

Nc1cc(-c2cccc3ccccc23)nc(N)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.49
HSP90AA1 P07900 3/20 0.49
HSP90AB1 P08238 2/20 0.49
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HTR1B P28222 1/20 0.43
HTR2B P41595 1/20 0.43
GPR65 Q8IYL9 1/20 0.43
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPK10 P53779 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALOX15 P16050 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
CCNT1 O60563 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5749719 0.98 DHFR (0.47) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL29861015 0.89 HSP90AA1 (0.51) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL5750835 0.83 MEN1 (0.48) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL5748593 0.83 ADORA2A (0.67) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL5746670 0.83 HSP90AA1 (0.60) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL5749587 0.83 HSP90AA1 (0.73) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL8329880 0.81 HSP90AA1 (0.59) DHFRHSP90AA1HSP90AB1MEN1KMT2A
Hydrochloric Acid SCHEMBL5748225 0.81 HSP90AA1 (0.71) DHFRHSP90AA1HSP90AB1MEN1KMT2A
SCHEMBL8328709 0.81 HSP90AA1 (0.71) DHFRHSP90AA1HSP90AB1MEN1KMT2A
Hydrochloric Acid SCHEMBL5749835 0.81 ADORA2A (0.65) DHFRHSP90AA1HSP90AB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP claimed
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed