SCHEMBL7377904

SCHEMBL7377904

COc1ccc(NC(c2ccc(Cl)cc2CN2CCC[C@]2(C(N)=O)C(=O)OC(C)(C)C)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.35
DDR1 Q08345 1/20 0.34
MGLL Q99685 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KCNH2 Q12809 1/20 0.32
EP300 Q09472 2/20 0.32
CREBBP Q92793 2/20 0.32
S1PR1 P21453 1/20 0.32
P2RX3 P56373 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378447 0.90 MDM2 (0.35) MDM2DDR1MEN1KMT2AL3MBTL1
SCHEMBL7379279 0.85 CNR1 (0.35) MDM2DDR1ALDH1A1EP300CREBBP
SCHEMBL7379415 0.84 MAPT (0.32) MDM2DDR1MGLLMEN1KMT2A
SCHEMBL6925564 0.76 EGFR (0.45) MDM2DDR1KDM4EALDH1A1EP300
SCHEMBL6924610 0.72 ALDH1A1 (0.61) MEN1KMT2AALDH1A1EP300CREBBP
SCHEMBL6926419 0.72 MEN1 (0.48) MDM2MEN1KMT2AL3MBTL1KDM4E
SCHEMBL6923255 0.66 HTR2C (0.46) MDM2DDR1KDM4EALDH1A1
SCHEMBL6926479 0.64 F2 (0.60) MEN1KMT2AALDH1A1EP300CREBBP
SCHEMBL6925575 0.64 EGFR (0.45) MDM2KDM4EALDH1A1EP300CREBBP
SCHEMBL6919944 0.62 HTRA1 (0.42) DDR1MEN1KMT2AL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002050056-A1 BENZYLAMINE DERIVATIVES AND THEIR USE AS THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-06-27 WO disclosed