SCHEMBL7378185

SCHEMBL7378185

N=C(N)Nc1cccc(C(=O)Nc2ccc(CC(NC(=O)c3ccccc3)C(=O)O)cc2)c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.57
ITGA2B P08514 9/20 0.57
ITGAV P06756 7/20 0.57
ITGB1 P05556 6/20 0.57
ITGB5 P18084 6/20 0.57
ACE P12821 2/20 0.50
GPR132 Q9UNW8 1/20 0.50
MMP9 P14780 1/20 0.50
PTPN1 P18031 2/20 0.49
POLB P06746 1/20 0.49
KMT2A Q03164 1/20 0.49
F10 P00742 2/20 0.49
AGTR2 P50052 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378190 1.00 ITGB3 (0.57) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL8058939 0.91 PTPN1 (0.57) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7377326 0.91 ITGB1 (0.70) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7377320 0.91 ITGB1 (0.70) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL18068435 0.89 ITGB1 (0.63) ITGB1
SCHEMBL7376050 0.89 ITGB3 (0.61) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7376058 0.89 ITGB3 (0.61) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7380048 0.88 NPC1 (0.53) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7380047 0.88 NPC1 (0.53) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7372900 0.88 ITGB3 (0.56) ITGB3ITGA2BITGAVITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-B1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2002-02-06 EP claimed
EP-1157985-A1 Para- substituted phenylene derivatives and their use as integrin antagonists G.D. SEARLE & CO. (US) 2001-11-28 EP claimed
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0891325-B1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2002-02-06 EP disclosed
US-6251944-B1 (VITRONECTIN RECEPTOR) INTEGRIN ANTAGONIST, USEFUL FOR TREATING ANGIOGENESIS, TUMOR GROWTH, TUMOR METASTASIS, OSTEOPOROSIS AND HUMORAL HYPERCALCEMIA OF MALIGNANCY G. D. SEARLE & COMPANY 2001-06-26 US disclosed