SCHEMBL7378337

SCHEMBL7378337

NN=CNc1cccc(C(=O)Nc2ccc(CCC(=O)O)cc2-c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.46
ITGA2B P08514 2/20 0.46
ITGB1 P05556 1/20 0.46
ITGAV P06756 1/20 0.46
ITGB5 P18084 1/20 0.46
NR1H4 Q96RI1 6/20 0.44
FFAR1 O14842 2/20 0.43
PPARG P37231 3/20 0.42
PPARD Q03181 3/20 0.42
PPARA Q07869 2/20 0.42
HSPH1 Q92598 1/20 0.42
HDAC1 Q13547 2/20 0.41
PLA2G10 O15496 1/20 0.41
PLA2G2A P14555 1/20 0.41
SLCO1B1 Q9Y6L6 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SIRT1 Q96EB6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378125 0.88 ITGB3 (0.47) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7378327 0.87 ITGB3 (0.54) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7861974 0.84 ITGB3 (0.64) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7373424 0.84 ITGB3 (0.64) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7373860 0.81 PTGER1 (0.44) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7378811 0.80 PTGER4 (0.48) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7379916 0.79 PPARG (0.51) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7452332 0.79 PPARG (0.63) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL7856525 0.78 PPARG (0.59) ITGB3ITGA2BITGB1ITGAVITGB5
SCHEMBL8371225 0.78 ITGB3 (0.53) ITGB3ITGA2BITGB1ITGAVITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP disclosed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed