SCHEMBL7378628

SCHEMBL7378628

Cc1cc(NC(=O)c2cccc(NC=NN)c2)ccc1CCC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.55
ITGB3 P05106 7/20 0.53
ITGA2B P08514 7/20 0.53
ITGAV P06756 6/20 0.53
ITGB1 P05556 3/20 0.47
ITGB5 P18084 3/20 0.47
KMT2A Q03164 5/20 0.46
POLB P06746 2/20 0.46
NR1H4 Q96RI1 2/20 0.43
MEN1 O00255 3/20 0.43
FFAR1 O14842 2/20 0.43
KCNK3 O14649 2/20 0.43
KCNK9 Q9NPC2 2/20 0.43
TP53 P04637 1/20 0.43
GLA P06280 1/20 0.43
FKBP5 Q13451 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380126 0.90 ITGB3 (0.53) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7376564 0.88 ITGB3 (0.67) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7379952 0.87 ITGB3 (0.48) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7378623 0.86 SMN1; SMN2 (0.58) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7508102 0.85 ITGB3 (0.48) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7861974 0.84 ITGB3 (0.64) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7373424 0.84 ITGB3 (0.64) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7378811 0.82 PTGER4 (0.48) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7380550 0.80 ITGB3 (0.43) SMN1; SMN2ITGB3ITGA2BITGAVITGB1
SCHEMBL7380190 0.79 KCNK3 (0.46) SMN1; SMN2ITGB3ITGA2BITGAVITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP disclosed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed