SCHEMBL7379673

SCHEMBL7379673

CCCc1nc2ccccc2n1Cc1ccc(-c2cscc2-c2nnn[nH]2)cc1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 12/20 0.56
AGTR1 P30556 4/20 0.53
AGTR2 P50052 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386011 0.94 AGTR1 (0.61) PPARGAGTR1AGTR2
SCHEMBL9194632 0.90 PPARG (0.62) PPARGAGTR1AGTR2
SCHEMBL7391199 0.85 PPARG (0.54) PPARGAGTR1AGTR2
SCHEMBL7389075 0.85 PPARG (0.52) PPARGAGTR1AGTR2
SCHEMBL8393351 0.85 AGTR1 (0.70) PPARGAGTR1AGTR2
SCHEMBL9194965 0.84 AGTR1 (0.66) PPARGAGTR1AGTR2
SCHEMBL9638103 0.84 PPARG (0.53) PPARGAGTR1AGTR2
SCHEMBL7383964 0.83 PPARG (0.54) PPARGAGTR1AGTR2
SCHEMBL8971427 0.83 PPARG (0.52) PPARGAGTR1AGTR2
SCHEMBL9031623 0.81 AGTR1 (0.56) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5177074-A Heterocyclic nitrogen compounds used to treat hypertension, cognitive dysfunction, anxiety or depression MERCK & CO., INC. (US) 1993-01-05 US disclosed
EP-0513979-A1 Angiotensin II antagonists incorporating a substituted thiophene or furan MERCK & CO. INC. (US) 1992-11-19 EP disclosed