SCHEMBL7379690

SCHEMBL7379690

CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)C(O)C(Cc1ccccc1)NC(=O)[C@H](Cc1cscn1)NC(=O)OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.57
ADORA2A P29274 1/20 0.57
ADORA2B P29275 1/20 0.57
ADORA1 P30542 1/20 0.57
KLK5 Q9Y337 1/20 0.47
ACE P12821 3/20 0.45
REN P00797 8/20 0.45
SCN9A Q15858 1/20 0.44
CTSD P07339 5/20 0.43
CTSE P14091 5/20 0.43
BACE1 P56817 5/20 0.43
CMA1 P23946 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7379695 1.00 ADORA3 (0.57) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7384427 0.91 ADORA3 (0.65) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7384430 0.91 ADORA3 (0.65) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7380113 0.88 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7380116 0.88 ADORA3 (0.58) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7387622 0.88 ADORA3 (0.64) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7387620 0.88 ADORA3 (0.64) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7383993 0.86 KLK5 (0.61) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7383991 0.86 KLK5 (0.61) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7383340 0.86 ADORA3 (0.76) ADORA3ADORA2AADORA2BADORA1KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498680-A1 New beta-amino-alpha-hydroxycarboxylic acids and their use Sankyo Company Limited (JP) 1992-08-12 EP disclosed