SCHEMBL7380663

SCHEMBL7380663

CC(C)=CCN(c1ccc(C(C)C)cc1)C1CCN(CCC(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 10/20 0.45
CCR5 P51681 3/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KCNA3 P22001 1/20 0.35
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7391056 0.93 CACNA1B (0.43) CACNA1BCCR5OPRM1OPRL1ALDH1A1
SCHEMBL7387556 0.87 CACNA1B (0.42) CACNA1BCCR5ALDH1A1MAOB
SCHEMBL7389238 0.86 CACNA1B (0.41) CACNA1BOPRM1ALDH1A1MAOB
SCHEMBL7381981 0.86 CACNA1B (0.49) CACNA1BCCR5NOS3NOS1NOS2
SCHEMBL7421570 0.83 CACNA1B (0.43) CACNA1BCCR5ALDH1A1MAOB
SCHEMBL7385467 0.83 CACNA1B (0.49) CACNA1BCCR5OPRM1
SCHEMBL7390855 0.82 CACNA1B (0.44) CACNA1BCCR5OPRM1OPRL1
SCHEMBL7384735 0.81 CACNA1B (0.43) CACNA1BALDH1A1
SCHEMBL7383857 0.81 ALDH1A1 (0.44) CACNA1BALDH1A1
SCHEMBL7389836 0.81 CACNA1B (0.69) CACNA1BCCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251919-B1 ADMINISTERING ANILINE DERIVATIVE FOR THERAPY OF PAIN WARNER-LAMBERT 2001-06-26 US claimed
WO-1999043658-A1 HETEROCYCLIC SUBSTITUTED ANILINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1999-09-02 WO claimed
US-6251919-B1 ADMINISTERING ANILINE DERIVATIVE FOR THERAPY OF PAIN WARNER-LAMBERT 2001-06-26 US disclosed
WO-1999043658-A1 HETEROCYCLIC SUBSTITUTED ANILINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1999-09-02 WO disclosed