SCHEMBL7380944

SCHEMBL7380944

CCOC(=O)C(C)(Cc1ccc(SC)cc1)C(=O)OCC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 2/20 0.55
ALDH1A1 P00352 5/20 0.43
TSHR P16473 4/20 0.43
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
HSD17B10 Q99714 1/20 0.43
MAPT P10636 2/20 0.42
RECQL P46063 1/20 0.41
EPHX2 P34913 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.38
OPRK1 P41145 1/20 0.38
ABCB11 O95342 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15905970 0.89 MMP8 (0.56) MMP8ALDH1A1TSHRLMNARECQL
SCHEMBL28737716 0.83 MMP8 (0.60) MMP8ALDH1A1TSHRLMNAMAPT
SCHEMBL7362869 0.82 MMP8 (0.59) MMP8ALDH1A1TSHRLMNAMAPT
SCHEMBL2370973 0.82 MMP8 (0.59) MMP8ALDH1A1TSHRKDM4ELMNA
SCHEMBL28753087 0.81 MMP8 (0.57) MMP8ALDH1A1KDM4ELMNAMAPT
SCHEMBL458395 0.81 MMP8 (0.57) MMP8ALDH1A1TSHRLMNARECQL
SCHEMBL8710582 0.80 MMP8 (0.79) MMP8ALDH1A1TSHRLMNAHSD17B10
SCHEMBL24733330 0.79 MMP8 (0.56) MMP8ALDH1A1TSHRKDM4ELMNA
SCHEMBL7383887 0.78 EPHX2 (0.45) TSHRKDM4EMAPTEPHX2NR1H4
SCHEMBL12142745 0.78 MMP8 (0.55) MMP8ALDH1A1TSHRLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208240-A Alzeheimer's, cardiovascular, respiratory MERRELL DOW PHARMACEUTICALS INC. (US) 1993-05-04 US disclosed
EP-0503563-A2 Novel 8-substituted purines as selective adenosine receptor agents MERRELL PHARMACEUTICALS INC. (US) 1992-09-16 EP disclosed