SCHEMBL7384289

SCHEMBL7384289

O=C(Nc1ccc2nccnc2c1)c1c[nH]c2c1C(=O)CCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.44
RAB9A P51151 9/20 0.44
SMN1; SMN2 Q16637 8/20 0.44
ALDH1A1 P00352 7/20 0.44
KDM4E B2RXH2 6/20 0.44
HPGD P15428 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
KLK7 P49862 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
KMT2A Q03164 8/20 0.40
MAPT P10636 7/20 0.40
TP53 P04637 5/20 0.40
GAA P10253 3/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387328 0.87 NPC1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL7366686 0.81 SNCA (0.46) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL7384705 0.81 BUB1 (0.43) ALDH1A1KDM4EPOLBHTTBUB1
SCHEMBL7364883 0.80 LMNA (0.46) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL7397306 0.79 MAPT (0.45) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL5736172 0.79 CFTR (0.59) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL5734680 0.79 CFTR (0.48) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL7360138 0.79 LMNA (0.43) NPC1RAB9ASMN1; SMN2KDM4EHPGD
SCHEMBL7397449 0.79 MAPT (0.47) SMN1; SMN2ALDH1A1KDM4EKMT2AMAPT
SCHEMBL7397423 0.79 NPC1 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723462-A SLEEP AND SEIZURE DISORDERS; COGNITION ACTIVATORS, ANXIOLYTIC AGENTS NEUROGEN CORPORATION (US) 1998-03-03 US claimed
US-6096887-A USEFUL IN THE DIAGNOSIS AND TREATMENT OF ANXIETY, SLEEP AND SEIZURE DISORDERS, OVERDOSE WITH BENZODIAZEPINE DRUGS AND FOR ENHANCEMENT OF MEMORY. NEUROGEN CORPORATION (US) 2000-08-01 US disclosed
US-5723462-A SLEEP AND SEIZURE DISORDERS; COGNITION ACTIVATORS, ANXIOLYTIC AGENTS NEUROGEN CORPORATION (US) 1998-03-03 US disclosed
WO-1998002433-A1 CERTAIN FUSED PYRROLECARBOXAMIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO disclosed