SCHEMBL7384792

SCHEMBL7384792

CCOC(=O)C(Cc1coc2cc(C#N)ccc12)c1ccc(O[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.49
ALK Q9UM73 1/20 0.42
CETP P11597 1/20 0.38
F10 P00742 8/20 0.37
F2 P00734 5/20 0.37
PRSS1 P07477 3/20 0.37
PRSS2 P07478 3/20 0.37
PRSS3 P35030 3/20 0.37
PLG P00747 2/20 0.37
ALDH2 P05091 1/20 0.36
USP30 Q70CQ3 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384790 0.94 GPR119 (0.49) GPR119ALKCETPF10F2
SCHEMBL7384317 0.87 GPR119 (0.49) GPR119ALKCETPF10F2
SCHEMBL7386798 0.85 GPR119 (0.50) GPR119ALKCETPF10F2
SCHEMBL7389231 0.85 GPR119 (0.54) GPR119ALKCETPF10F2
SCHEMBL7386795 0.84 GPR119 (0.49) GPR119ALKCETPF10F2
SCHEMBL7384314 0.84 F10 (0.51) GPR119ALKCETPF10F2
SCHEMBL6928672 0.83 GPR119 (0.53) GPR119ALKCETPF10F2
SCHEMBL6925447 0.83 GPR119 (0.53) GPR119ALKCETPF10F2
SCHEMBL7388717 0.83 GPR119 (0.53) GPR119ALKCETPF10F2
SCHEMBL7385828 0.82 GPR119 (0.50) GPR119ALKCETPF10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620991-A ANTICOAGULANTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-04-15 US disclosed
US-5576343-A ANTICOAGULANTS; BLOOD-COAGULATION FACTOR X INHIBITORS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-11-19 US disclosed
EP-0540051-B1 Aromatic amidine derivatives and salts thereof DAIICHI SEIYAKU CO (JP) 1996-04-03 EP disclosed
EP-0540051-A1 Aromatic amidine derivatives and salts thereof DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-05-05 EP disclosed