SCHEMBL7386941

SCHEMBL7386941

c1ccc(CN2CC3CCCCC3(Cc3ccccc3)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.49
SLC6A4 P31645 3/20 0.49
SLC6A3 Q01959 3/20 0.49
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRM2 P08172 2/20 0.40
CHRM3 P20309 2/20 0.40
FUCA1 P04066 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386938 1.00 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL21480154 0.88 ALDH1A1 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL21480155 0.88 ALDH1A1 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL19779412 0.88 ALDH1A1 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL5654095 0.83 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5465323 0.83 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL20895733 0.79 CYP1A2 (0.42) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL16054301 0.79 CYP1A2 (0.42) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL8570353 0.79 CYP1A2 (0.42) SLC6A2SLC6A4SLC6A3ALDH1A1CYP1A2
SCHEMBL8388967 0.77 FUCA1 (0.44) ALDH1A1FUCA1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409929-A Treating psychosis, dyskinesia THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-25 US disclosed
EP-0626947-A1 HYDROISOINDOLINES AND HYDROISOQUINOLINES AS PSYCHOTROPIC DRUGS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-12-07 EP disclosed
WO-1993016047-A1 HYDROISOINDOLINES AND HYDROISOQUINOLINES AS PSYCHOTROPIC DRUGS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-08-19 WO disclosed
US-5216018-A Antidyskinetic agents DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-06-01 US disclosed