SCHEMBL738710

SCHEMBL738710

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)N(C(=O)O)C(C)(C)C)C2)nc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.37
HRH1 P35367 4/20 0.37
CYP2D6 P10635 3/20 0.37
TACR1 P25103 6/20 0.35
CASR P41180 2/20 0.35
CHRM1 P11229 1/20 0.34
CTNNB1 P35222 1/20 0.32
MAPT P10636 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
F2 P00734 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL744560 0.95 HRH1 (0.37) KCNH2HRH1CYP2D6TACR1CASR
SCHEMBL742065 0.91 HRH1 (0.39) KCNH2HRH1CYP2D6TACR1CHRM1
SCHEMBL738741 0.91 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1MAPT
SCHEMBL741317 0.91 HRH1 (0.45) KCNH2HRH1CYP2D6CHRM1PROKR1
SCHEMBL740611 0.90 KCNH2 (0.38) KCNH2HRH1CYP2D6CHRM1CTNNB1
SCHEMBL740359 0.89 ADORA2A (0.40) KCNH2HRH1CYP2D6TACR1CASR
SCHEMBL739969 0.88 DPP4 (0.37) KCNH2HRH1CYP2D6TACR1CASR
SCHEMBL739968 0.88 DPP4 (0.37) KCNH2HRH1CYP2D6TACR1CASR
SCHEMBL742192 0.86 HRH1 (0.40) KCNH2HRH1CYP2D6CHRM1MAPT
SCHEMBL762582 0.85 CASR (0.37) KCNH2HRH1CYP2D6TACR1CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed