SCHEMBL744560

SCHEMBL744560

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)N(C(=O)O)C(C)(C)C)C2)nc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.37
KCNH2 Q12809 3/20 0.37
CYP2D6 P10635 2/20 0.37
OPRM1 P35372 1/20 0.36
TACR1 P25103 5/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CASR P41180 2/20 0.35
CHRM1 P11229 1/20 0.34
ITK Q08881 1/20 0.33
GNRHR P30968 1/20 0.33
CNR2 P34972 3/20 0.33
KMT2A Q03164 1/20 0.33
BCHE P06276 1/20 0.32
CNR1 P21554 1/20 0.32
CTNNB1 P35222 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL738710 0.95 KCNH2 (0.37) HRH1KCNH2CYP2D6TACR1ALDH1A1
SCHEMBL741317 0.91 HRH1 (0.45) HRH1KCNH2CYP2D6CHRM1
SCHEMBL742192 0.90 HRH1 (0.40) HRH1KCNH2CYP2D6CHRM1ITK
SCHEMBL763214 0.88 OPRM1 (0.39) HRH1KCNH2CYP2D6OPRM1ALDH1A1
SCHEMBL738741 0.87 KCNH2 (0.39) HRH1KCNH2CYP2D6ALDH1A1LMNA
SCHEMBL742065 0.87 HRH1 (0.39) HRH1KCNH2CYP2D6TACR1CHRM1
SCHEMBL740611 0.86 KCNH2 (0.38) HRH1KCNH2CYP2D6CHRM1CTNNB1
SCHEMBL762655 0.85 CASR (0.37) HRH1KCNH2CYP2D6OPRM1TACR1
SCHEMBL740359 0.85 ADORA2A (0.40) HRH1KCNH2CYP2D6TACR1CASR
SCHEMBL742487 0.84 HRH1 (0.36) HRH1KCNH2CYP2D6TACR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed