SCHEMBL7387992

SCHEMBL7387992

Brc1csc(Br)n1.Brc1csc(C#Cc2ccccc2)n1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 12/20 0.60
APP P05067 1/20 0.41
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313419 0.95 GRM5 (0.66) GRM5APPCHEK1
SCHEMBL1656957 0.75 GRM5 (0.58) GRM5CHEK1
SCHEMBL15692608 0.72 GRM5 (0.55) GRM5APPCHEK1
SCHEMBL67456 0.72
SCHEMBL1656880 0.69 TDP1 (0.59) GRM5CHEK1
SCHEMBL24075982 0.68 GRM5 (0.54) GRM5APPCHEK1
SCHEMBL1656990 0.67 GRM5 (0.52) GRM5CHEK1
SCHEMBL1657308 0.67 GRM5 (0.52) GRM5CHEK1
SCHEMBL21189528 0.66 GRM5 (0.33) GRM5
SCHEMBL15322434 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed