SCHEMBL7388449

SCHEMBL7388449

CCCCOc1ccc([S+]([O-])N2CCN(C)CC2)cc1-c1nc2c([nH]1)c(=O)[nH]c(=O)n2CCC

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 16/20 0.61
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GLA P06280 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ADORA2A P29274 3/20 0.45
ADORA2B P29275 3/20 0.45
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5827741 0.83 PDE5A (0.88) PDE5APDE3BPDE3A
SCHEMBL5827328 0.79 PDE5A (0.89) PDE5A
SCHEMBL5827664 0.77 PDE5A (0.74) PDE5AADORA2AADORA2B
SCHEMBL5827847 0.76 PDE5A (0.84) PDE5A
SCHEMBL2562501 0.76 PDE5A (0.69) PDE5A
SCHEMBL5827707 0.73 PDE5A (0.77) PDE5A
SCHEMBL5827475 0.73 PDE5A (0.75) PDE5A
SCHEMBL7035902 0.71 PDE5A (0.51) PDE5AKDM4EKMT2AADORA2APDE3B
SCHEMBL7003278 0.69 PDE5A (0.71) PDE5AKDM4EALDH1A1KMT2AADORA2A
SCHEMBL5827900 0.69 PDE5A (0.65) PDE5APDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1198464-A1 8-PHENYL-6,9-DIHYDRO- 1,2,4]TRIAZOLO 3,4- i i /i ]PURIN-5-ONE DERIVATIVES Almirall Prodesfarma, S.A. (ES) 2002-04-24 EP disclosed
WO-2001007441-A1 8-PHENYL-6,9-DIHYDRO-[1,2,4]TRIAZOLO[3,4-i]PURIN-5-ONE DERIVATIVES ALMIRALL PRODESFARMA S.A. (ES) 2001-02-01 WO disclosed