SCHEMBL739173

SCHEMBL739173

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc(C(=O)N5CCOCC5)cc4)cc3)C2)nc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.47
HTR2B P41595 1/20 0.43
KCNH2 Q12809 6/20 0.43
PTGER4 P35408 1/20 0.41
CYP2D6 P10635 2/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CB P42338 1/20 0.40
PROKR1 Q8TCW9 1/20 0.39
HRH3 Q9Y5N1 5/20 0.39
CHRM1 P11229 2/20 0.39
CHRM2 P08172 1/20 0.39
ADRA2C P18825 1/20 0.39
CHRM3 P20309 1/20 0.39
DRD4 P21917 1/20 0.39
SLC6A2 P23975 1/20 0.39
HRH2 P25021 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739174 1.00 HRH1 (0.47) HRH1HTR2BKCNH2PTGER4CYP2D6
SCHEMBL741193 0.92 HRH1 (0.46) HRH1KCNH2CYP2D6PIK3CDPIK3CB
SCHEMBL741194 0.92 HRH1 (0.46) HRH1KCNH2CYP2D6PIK3CDPIK3CB
SCHEMBL740879 0.91 HTR2B (0.43) HRH1HTR2BKCNH2CYP2D6PROKR1
SCHEMBL740878 0.91 HTR2B (0.43) HRH1HTR2BKCNH2CYP2D6PROKR1
SCHEMBL738819 0.90 HRH1 (0.43) HRH1HTR2BKCNH2CYP2D6CHRM1
SCHEMBL738820 0.90 HRH1 (0.43) HRH1HTR2BKCNH2CYP2D6CHRM1
SCHEMBL738739 0.90 HRH1 (0.46) HRH1HTR2BKCNH2CYP2D6CHRM1
SCHEMBL738740 0.90 HRH1 (0.46) HRH1HTR2BKCNH2CYP2D6CHRM1
SCHEMBL740626 0.90 HRH1 (0.42) HRH1HTR2BKCNH2CYP2D6PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed