SCHEMBL740878

SCHEMBL740878

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc(C(=O)N5CC[C@@H](O)C5)cc4)cc3)C2)nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.43
PROKR1 Q8TCW9 3/20 0.41
HRH1 P35367 5/20 0.40
CYP2D6 P10635 4/20 0.40
KCNH2 Q12809 6/20 0.40
HRH3 Q9Y5N1 8/20 0.40
CHRM1 P11229 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740879 1.00 HTR2B (0.43) HTR2BPROKR1HRH1CYP2D6KCNH2
SCHEMBL739173 0.91 HRH1 (0.47) HTR2BPROKR1HRH1CYP2D6KCNH2
SCHEMBL739174 0.91 HRH1 (0.47) HTR2BPROKR1HRH1CYP2D6KCNH2
SCHEMBL738819 0.90 HRH1 (0.43) HTR2BHRH1CYP2D6KCNH2CHRM1
SCHEMBL738820 0.90 HRH1 (0.43) HTR2BHRH1CYP2D6KCNH2CHRM1
SCHEMBL738740 0.90 HRH1 (0.46) HTR2BHRH1CYP2D6KCNH2CHRM1
SCHEMBL738739 0.90 HRH1 (0.46) HTR2BHRH1CYP2D6KCNH2CHRM1
SCHEMBL740626 0.90 HRH1 (0.42) HTR2BPROKR1HRH1CYP2D6KCNH2
SCHEMBL740625 0.90 HRH1 (0.42) HTR2BPROKR1HRH1CYP2D6KCNH2
SCHEMBL739379 0.89 HRH1 (0.44) PROKR1HRH1CYP2D6KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed