SCHEMBL739358

SCHEMBL739358

COCCCn1c(C2CCCNC2)nc2ccc(C#N)cc21

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.53
HRH1 P35367 2/20 0.53
ADORA2A P29274 3/20 0.42
BRD4 O60885 3/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
REN P00797 1/20 0.40
ITK Q08881 6/20 0.40
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 2/20 0.39
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739357 1.00 CHRM1 (0.53) CHRM1HRH1ADORA2ABRD4DRD2
SCHEMBL737976 0.86 HRH1 (0.55) CHRM1HRH1BRD4RENOPRM1
SCHEMBL740755 0.86 HRH1 (0.52) CHRM1HRH1BRD4RENOPRM1
SCHEMBL740756 0.86 HRH1 (0.52) CHRM1HRH1BRD4RENOPRM1
SCHEMBL742773 0.86 HRH1 (0.54) CHRM1HRH1BRD4RENOPRM1
SCHEMBL737977 0.86 HRH1 (0.55) CHRM1HRH1BRD4RENOPRM1
SCHEMBL742774 0.86 HRH1 (0.54) CHRM1HRH1BRD4RENOPRM1
SCHEMBL739843 0.84 HRH1 (0.70) CHRM1HRH1BRD4RENOPRM1
SCHEMBL739842 0.84 HRH1 (0.70) CHRM1HRH1BRD4RENOPRM1
SCHEMBL740511 0.82 CHRM1 (0.48) CHRM1HRH1ADORA2ABRD4REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed