SCHEMBL739437

SCHEMBL739437

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccc(C(=O)NCCO)c(F)c4)cc3)NC(=O)O)C2)nc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 9/20 0.40
CYP2D6 P10635 7/20 0.40
MAPK1 P28482 6/20 0.39
KCNH2 Q12809 8/20 0.38
CHRM1 P11229 3/20 0.38
CHRM4 P08173 1/20 0.37
ROCK2 O75116 1/20 0.36
RPS6KA5 O75582 1/20 0.36
RPS6KA4 O75676 1/20 0.36
PRKACA P17612 1/20 0.36
GSK3B P49841 1/20 0.36
PRKX P51817 1/20 0.36
LIMK1 P53667 1/20 0.36
ROCK1 Q13464 1/20 0.36
PRKG1 Q13976 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742610 0.96 HRH1 (0.41) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL16301226 0.92 HRH1 (0.38) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL762743 0.92 HRH1 (0.41) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL740525 0.92 HRH1 (0.41) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL740524 0.92 HRH1 (0.41) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL744675 0.89 HRH1 (0.40) HRH1CYP2D6KCNH2CHRM1
SCHEMBL10293052 0.89 HRH1 (0.39) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL740088 0.89 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1
SCHEMBL763245 0.88 HRH1 (0.42) HRH1CYP2D6MAPK1KCNH2CHRM1
SCHEMBL740424 0.88 HRH1 (0.41) HRH1CYP2D6MAPK1KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed