SCHEMBL739666

SCHEMBL739666

COCCCn1c(C2CCCN(C(=O)CC(N)Cc3ccc4ccccc4c3)C2)nc2ccc(C(C)C)cc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.39
HRH1 P35367 7/20 0.39
CYP2D6 P10635 5/20 0.39
CHRM1 P11229 3/20 0.38
PPARA Q07869 1/20 0.37
CYP3A4 P08684 1/20 0.36
PROKR1 Q8TCW9 4/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
ADORA2A P29274 1/20 0.34
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34
ITGAL P20701 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762659 1.00 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1PPARA
SCHEMBL739665 1.00 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1PPARA
SCHEMBL763459 0.94 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1PPARA
SCHEMBL739989 0.94 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1PPARA
SCHEMBL739988 0.94 KCNH2 (0.39) KCNH2HRH1CYP2D6CHRM1PPARA
SCHEMBL740604 0.92 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL738317 0.92 HRH1 (0.39) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL740603 0.92 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL739244 0.92 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL739245 0.92 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed