SCHEMBL740604

SCHEMBL740604

COCCCn1c(C2CCCN(C(=O)CC(N)Cc3ccc4ccccc4c3)C2)nc2ccc(OC)cc21

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.43
CYP3A4 P08684 1/20 0.41
HRH1 P35367 6/20 0.39
CYP2D6 P10635 4/20 0.39
CHRM1 P11229 3/20 0.38
ALDH1A1 P00352 4/20 0.37
LMNA P02545 2/20 0.37
TSHR P16473 2/20 0.37
RAB9A P51151 1/20 0.37
HTT P42858 1/20 0.37
MAPT P10636 3/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPK10 P53779 1/20 0.36
NMT2 O60551 1/20 0.36
NMT1 P30419 1/20 0.36
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740603 1.00 KCNH2 (0.43) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL738317 0.93 HRH1 (0.39) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739244 0.93 HRH1 (0.46) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739245 0.93 HRH1 (0.46) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL762659 0.92 KCNH2 (0.39) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739991 0.92 HRH1 (0.44) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL742135 0.92 KCNH2 (0.39) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739990 0.92 HRH1 (0.44) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739666 0.92 KCNH2 (0.39) KCNH2CYP3A4HRH1CYP2D6CHRM1
SCHEMBL739665 0.92 KCNH2 (0.39) KCNH2CYP3A4HRH1CYP2D6CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed