SCHEMBL7397256

SCHEMBL7397256

COC(=O)[C@@H](N)Cc1ccc(N(C(=O)OCc2ccccc2)C(=O)C2CCNCC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.43
ITGA2B P08514 5/20 0.43
LTA4H P09960 1/20 0.39
CTSD P07339 2/20 0.39
ITGAV P06756 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
TYR P14679 1/20 0.39
SLC15A1 P46059 1/20 0.39
ABCB1 P08183 1/20 0.38
TSHR P16473 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
ENPP2 Q13822 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5162805 0.78 ITGB1 (0.51)
Hydrochloric Acid SCHEMBL7527724 0.76 LTA4H (0.41) LTA4HKDM1AMAOASLC15A1ABCB1
Phenylalanine Methyl Ester SCHEMBL74888 0.71 SLC7A5 (0.63) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL27880854 0.71 SLC7A5 (0.63) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL74887 0.71 SLC7A5 (0.63) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL186022 0.71 SLC7A5 (0.63) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL136409 0.70 SLC7A5 (0.61) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL2237414 0.70 SLC7A5 (0.61) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL2728392 0.70 SLC7A5 (0.61) LTA4HSLC15A1ALDH1A1
Phenylalanine Methyl Ester SCHEMBL136408 0.70 SLC7A5 (0.61) LTA4HSLC15A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144435-A2 PYROGLUTAMIC ACID DERIVATIVES AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2001-10-17 EP disclosed
WO-2000043413-A2 PYROGLUTAMIC ACID DERIVATIVES AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2000-07-27 WO disclosed