SCHEMBL7398283

SCHEMBL7398283

COc1cccc(N2CCN(c3ccncc3)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.69
NPC1 O15118 2/20 0.69
ADRB1 P08588 1/20 0.61
KDM4E B2RXH2 2/20 0.59
GFER P55789 1/20 0.59
DRD2 P14416 1/20 0.59
KCNH2 Q12809 1/20 0.59
ROCK2 O75116 1/20 0.57
ALDH1A1 P00352 5/20 0.56
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
RAB9A P51151 2/20 0.55
KHK P50053 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
DHFR P00374 1/20 0.53
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11074672 0.88 ADRB1 (0.76) MAPTNPC1ADRB1KDM4EGFER
SCHEMBL19212406 0.86 ADRB1 (0.69) MAPTNPC1ADRB1KDM4EDRD2
SCHEMBL27371785 0.84 KDM4E (0.75) MAPTNPC1KDM4EGFERDRD2
SCHEMBL8890453 0.82 GAA (0.69) MAPTNPC1ADRB1DRD2ALDH1A1
SCHEMBL1372927 0.81 KCNH2 (0.69) MAPTNPC1ADRB1KDM4EDRD2
SCHEMBL23675047 0.80 ADRB1 (0.71) MAPTNPC1ADRB1KDM4EDRD2
SCHEMBL3051915 0.80 ADRB1 (0.71) MAPTNPC1ADRB1KDM4EDRD2
SCHEMBL30255158 0.80 ADRB1 (0.71) MAPTNPC1ADRB1KDM4EDRD2
SCHEMBL12526595 0.80 AOC3 (0.53) MAPTNPC1KDM4EGFERDRD2
SCHEMBL1365556 0.79 ADRB1 (0.65) MAPTNPC1ADRB1KDM4EGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed