SCHEMBL7398463

SCHEMBL7398463

Oc1ccc(N2CCN(CCC3OCCc4ccccc43)CC2)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.79
HTR2A P28223 7/20 0.79
DRD4 P21917 6/20 0.79
HTR1A P08908 5/20 0.79
ADRA2A P08913 1/20 0.79
ADRA2B P18089 1/20 0.79
ADRA2C P18825 1/20 0.79
DRD1 P21728 1/20 0.79
ADRA1D P25100 1/20 0.79
ADRA1A P35348 1/20 0.79
ADRA1B P35368 1/20 0.79
DRD3 P35462 1/20 0.79
HTR2B P41595 1/20 0.79
HTR1D P28221 8/20 0.74
CA12 O43570 1/20 0.72
CA1 P00915 1/20 0.72
CA2 P00918 1/20 0.72
CA4 P22748 1/20 0.72
CA6 P23280 1/20 0.72
CA5A P35218 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7404598 0.99 DRD2 (0.78) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL5698946 0.90 DRD2 (0.82) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL7402186 0.89 DRD2 (0.80) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7403359 0.88 DRD2 (0.79) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL5698997 0.88 DRD2 (1.00) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7400484 0.88 DRD2 (0.79) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL29366062 0.87 DRD2 (0.98) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL8179298 0.87 DRD2 (0.78) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL8170055 0.87 DRD2 (0.98) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL5698979 0.87 DRD2 (0.73) DRD2HTR2ADRD4HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737189-B1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS UPJOHN CO (US) 1999-07-28 EP claimed
EP-0737189-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1996-10-16 EP claimed
WO-1995018118-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS THE UPJOHN COMPANY (US) 1995-07-06 WO claimed