SCHEMBL7398486

SCHEMBL7398486

CCC[C@H](C[C@H](O[Si](C)(C)C(C)(C)C)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.44
ALDH1A1 P00352 2/20 0.43
ATM Q13315 1/20 0.43
ACE P12821 1/20 0.42
PSEN1 P49768 3/20 0.42
PSEN2 P49810 3/20 0.42
APH1B Q8WW43 3/20 0.42
NCSTN Q92542 3/20 0.42
APH1A Q96BI3 3/20 0.42
PSENEN Q9NZ42 3/20 0.42
APP P05067 1/20 0.42
CTSK P43235 3/20 0.41
CTSS P25774 2/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
REN P00797 3/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446803 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL6305846 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL7283432 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL5142842 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL7398818 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL7796450 0.92 KLK5 (0.47) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL7412747 0.90 BACE1 (0.43) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL9057406 0.89 PSEN1 (0.48) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL10337125 0.89 PSEN1 (0.48) KLK5ALDH1A1ATMACEPSEN1
SCHEMBL7404966 0.89 PSEN1 (0.48) KLK5ALDH1A1ATMACEPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610431-A1 HIV PROTEASE INHIBITORS CONTAINING GUANIDINE SMITHKLINE BEECHAM CORPORATION (US) 1994-08-17 EP disclosed
WO-1993009132-A1 HIV PROTEASE INHIBITORS CONTAINING GUANIDINE SMITHKLINE BEECHAM CORPORATION (US) 1993-05-13 WO disclosed