SCHEMBL7399086

SCHEMBL7399086

COC(=O)COc1ccc2nccc(N3CCN(c4ccncc4)CC3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.49
NCF1 P14598 1/20 0.49
GAA P10253 3/20 0.46
CDK8 P49336 3/20 0.43
MAPT P10636 2/20 0.43
METAP1 P53582 1/20 0.42
CCNC P24863 1/20 0.42
PDGFRB P09619 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HRH3 Q9Y5N1 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402500 0.88 METAP1 (0.51) NCF1GAACDK8MAPTMETAP1
SCHEMBL7398874 0.74 GAA (0.49) GAAMAPTITGB3ITGA2BALDH1A1
SCHEMBL7399938 0.74 SLC22A12 (0.56) SLC22A12GAAALDH1A1KDM4EMEN1
SCHEMBL7402704 0.73 GAA (0.48) GAAMAPTHRH3MEN1KMT2A
SCHEMBL7398918 0.73 POLB (0.60) HRH3
SCHEMBL7335436 0.73 HRH3 (0.59) MAPTITGB3ITGA2BALDH1A1HRH3
SCHEMBL7394056 0.73 TRPV1 (0.62) GAAMAPTPDGFRBALDH1A1MEN1
SCHEMBL7405234 0.73 GAA (0.50) GAAMAPTALDH1A1HRH3MEN1
SCHEMBL7405501 0.73 F10 (0.49) GAAMAPTITGB3ITGA2BALDH1A1
SCHEMBL7332909 0.73 ACACB (0.47) GAAMAPTITGB3ITGA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed