SCHEMBL739955

SCHEMBL739955

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)NC(=O)O)C2)nc2ccc(C#N)cc21

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.43
HRH1 P35367 2/20 0.39
KCNH2 Q12809 2/20 0.39
CYP2D6 P10635 1/20 0.39
ITK Q08881 10/20 0.38
CHRM1 P11229 1/20 0.38
PIN1 Q13526 1/20 0.38
TACR1 P25103 1/20 0.36
ALOX5AP P20292 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763244 0.92 ADORA2A (0.41) ADORA2AHRH1KCNH2CYP2D6ITK
SCHEMBL739252 0.91 KCNH2 (0.41) ADORA2AHRH1KCNH2CYP2D6CHRM1
SCHEMBL740708 0.91 HRH1 (0.39) ADORA2AHRH1KCNH2CYP2D6CHRM1
SCHEMBL739901 0.91 HRH1 (0.46) HRH1KCNH2CYP2D6CHRM1
SCHEMBL739752 0.90 ADORA2A (0.43) ADORA2AHRH1KCNH2CYP2D6ITK
SCHEMBL739753 0.90 ADORA2A (0.43) ADORA2AHRH1KCNH2CYP2D6ITK
SCHEMBL740857 0.90 KCNH2 (0.39) ADORA2AHRH1KCNH2CYP2D6ITK
SCHEMBL742275 0.90 HRH1 (0.42) ADORA2AHRH1KCNH2CYP2D6CHRM1
SCHEMBL740359 0.87 ADORA2A (0.40) ADORA2AHRH1KCNH2CYP2D6ITK
SCHEMBL741997 0.86 KCNH2 (0.35) HRH1KCNH2CYP2D6CHRM1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed