SCHEMBL763244

SCHEMBL763244

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)NC(=O)OC(C)(C)C)C2)nc2ccc(C#N)cc21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
ITK Q08881 9/20 0.36
CASR P41180 1/20 0.36
HRH1 P35367 3/20 0.36
KCNH2 Q12809 2/20 0.36
CYP2D6 P10635 1/20 0.36
REN P00797 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
CHRM1 P11229 1/20 0.35
HRH2 P25021 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739955 0.92 ADORA2A (0.43) ADORA2AITKHRH1KCNH2CYP2D6
SCHEMBL762577 0.91 CTSB (0.36) ADORA2ACTSBCTSSCTSKHRH1
SCHEMBL762648 0.91 HRH1 (0.36) ADORA2ACTSBCTSSCTSKHRH1
SCHEMBL762559 0.91 KCNH2 (0.39) CTSBCTSSCTSKHRH1KCNH2
SCHEMBL762785 0.91 HRH1 (0.42) CTSBCTSSCTSKHRH1KCNH2
SCHEMBL763206 0.91 HRH1 (0.40) CTSBCTSSCTSKHRH1KCNH2
SCHEMBL762513 0.91 KCNH2 (0.36) CTSBCTSSCTSKITKHRH1
SCHEMBL762657 0.91 PPARA (0.36) ADORA2ACTSBCTSSCTSKHRH1
SCHEMBL741447 0.90 ADORA2A (0.36) ADORA2ACTSBCTSSCTSKHRH1
SCHEMBL741446 0.90 ADORA2A (0.36) ADORA2ACTSBCTSSCTSKHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed