SCHEMBL7399740

SCHEMBL7399740

CCC(O)O.c1ccc(COCc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.65
CA1 P00915 4/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
TRPA1 O75762 1/20 0.47
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.45
HTT P42858 2/20 0.45
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
TACR1 P25103 2/20 0.43
IDO1 P14902 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isopropyl Alcohol SCHEMBL29076646 0.86 TSHR (0.71) TSHRCA1CA2CA7CA9
SCHEMBL29062355 0.86 TSHR (0.58) TSHRCA1CA2CA7CA9
Alcohol SCHEMBL9721767 0.84 TSHR (0.75) TSHRCA1CA2CA7CA9
Propane SCHEMBL11584021 0.84 TSHR (0.83) TSHRCA1CA2CA7CA9
Hydrogen Peroxide SCHEMBL28758135 0.83 TSHR (0.94) TSHRCA1CA2CA7CA9
SCHEMBL26087124 0.83 LMNA (0.62) TSHRCA1CA2CA7CA9
SCHEMBL4570490 0.82 CA1 (0.68) TSHRCA1CA2CA7CA9
SCHEMBL5516631 0.82 CA1 (0.68) TSHRCA1CA2CA7CA9
SCHEMBL2717725 0.82 CA1 (0.68) TSHRCA1CA2CA7CA9
SCHEMBL27713879 0.81 TSHR (0.52) TSHRCA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618926-B1 NEW PEPTIDE DERIVATIVES ASTRA AB (SE) 2000-03-01 EP disclosed
US-5955433-A DERIVATIVES OF B-CYCLOHEXYLALANINE-PROLINE-AGMATINE ARE ADMINISTERED AS ANTICOAGULANTS ASTRA AKTIEBOLAG (SE) 1999-09-21 US disclosed
US-5747460-A Method of treatment and prophylaxis of venous thrombosis ASTRA AKTIEBOLAG (SE) 1998-05-05 US disclosed
US-5736521-A ADMINISTERING AMINO ACID COMPOUND ASTRA AKTIEBOLAG (SE) 1998-04-07 US disclosed
US-5614499-A ANTICOAGULANTS; TREATMENT OR PROPHYLAXIS OF THROMBOSIS ASTRA AKTIEBOLAG (SE) 1997-03-25 US disclosed
EP-0618926-A1 NEW PEPTIDE DERIVATIVES Astra Aktiebolag (SE) 1994-10-12 EP disclosed
WO-1993011152-A1 NEW PEPTIDE DERIVATIVES AKTIEBOLAGET ASTRA (SE) 1993-06-10 WO disclosed