SCHEMBL7399801

SCHEMBL7399801

COC(=O)CCNC(=O)c1cccc(Br)n1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
HPGD P15428 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 1/20 0.49
GRM5 P41594 1/20 0.48
KDM5B Q9UGL1 1/20 0.41
PRSS1 P07477 1/20 0.41
CTSG P08311 1/20 0.41
CTRB1 P17538 1/20 0.41
CMA1 P23946 1/20 0.41
CTSA P10619 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14371962 0.82 ALDH1A1 (0.65) ALDH1A1HPGDSMN1; SMN2LMNAGRM5
SCHEMBL4088050 0.81 ALDH1A1 (0.60) ALDH1A1HPGDSMN1; SMN2LMNAGRM5
SCHEMBL8893000 0.80 CYP3A4 (0.55) ALDH1A1HPGDSMN1; SMN2LMNAGRM5
SCHEMBL3505447 0.79 ALDH1A1 (0.61) ALDH1A1HPGDLMNAGRM5CTSA
SCHEMBL10708175 0.79 ALDH1A1 (0.66) ALDH1A1HPGDLMNAGRM5CTSA
SCHEMBL1037003 0.79 ALDH1A1 (0.65) ALDH1A1HPGDSMN1; SMN2LMNAGRM5
SCHEMBL31055457 0.78 HPGD (0.57) ALDH1A1HPGDSMN1; SMN2LMNAGRM5
SCHEMBL6931 0.78 ALDH1A1 (0.57) ALDH1A1HPGDLMNAGRM5
SCHEMBL24150763 0.78 ALDH1A1 (0.60) ALDH1A1HPGDLMNAGRM5CTSA
Hydrochloric Acid SCHEMBL10707808 0.78 ALDH1A1 (0.60) ALDH1A1HPGDLMNAGRM5CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5563141-A INHIBIT CELL ADHESION FOR EXAMPLE, PLATELET AGGRE GATION ZENECA LIMITED (GB) 1996-10-08 US disclosed
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed