SCHEMBL7400258

SCHEMBL7400258

CCCc1cccc(NC2CCN(S(=O)(=O)c3ccc(CNC(=O)c4ccc(Cl)cc4)s3)CC2)c1.O=C(NCc1ccc(S(=O)(=O)N2CCC(Nc3cccc(C(F)(F)F)c3)CC2)s1)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 1/20 0.49
MAPK10 P53779 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 5/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CCR2 P41597 6/20 0.41
ACKR3 P25106 1/20 0.40
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
USP5 P45974 1/20 0.40
TP53 P04637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
TGM2 P21980 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1518735 0.94 MAPK9 (0.54) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2424312 0.93 MAPK9 (0.55) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2420821 0.88 MAPK9 (0.56) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2425499 0.87 MAPK9 (0.55) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2420483 0.85 MAPK9 (0.55) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL4189441 0.84 MAPK9 (0.57) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2421312 0.84 MAPK9 (0.57) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2422729 0.84 MAPK9 (0.57) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2422241 0.84 MEN1 (0.49) MAPK9MAPK10MEN1KMT2AMAPT
SCHEMBL2422037 0.84 MAPK9 (0.59) MAPK9MAPK10MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218374-A1 PHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2002-07-03 EP disclosed
WO-2001023378-A1 PHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-04-05 WO disclosed