SCHEMBL7400520

SCHEMBL7400520

CN(C)C(=O)Oc1ccc(CC(N)C(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.58
SLC7A5 Q01650 4/20 0.54
PTPN1 P18031 1/20 0.54
PTGS1 P23219 3/20 0.53
PKM P14618 2/20 0.53
ALPI P09923 1/20 0.53
XIAP P98170 1/20 0.53
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
ALDH1A1 P00352 3/20 0.49
KMT2A Q03164 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
LDHA P00338 1/20 0.49
ITGB1 P05556 2/20 0.48
ITGA4 P13612 2/20 0.48
CYP3A4 P08684 3/20 0.48
ALOX15 P16050 3/20 0.48
HIF1A Q16665 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TDP1 Q9NUW8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850501 1.00 RAB9A (0.58) RAB9ASLC7A5PTPN1PTGS1PKM
SCHEMBL31126214 0.86 SLC7A5 (0.59) SLC7A5PTPN1PTGS1PKMALPI
SCHEMBL8267901 0.85 RAB9A (0.54) RAB9APKMALDH1A1KMT2ANPSR1
SCHEMBL4843558 0.84 RAB9A (0.53) RAB9APKMALDH1A1KMT2ANPSR1
SCHEMBL22645606 0.84 SLC7A5 (0.61) SLC7A5PTPN1PTGS1PKMALPI
SCHEMBL671002 0.84 SLC7A5 (0.61) SLC7A5PTPN1PTGS1PKMALPI
SCHEMBL450849 0.84 SLC7A5 (0.61) SLC7A5PTPN1PTGS1PKMALPI
SCHEMBL2058791 0.83 RAB9A (0.51) RAB9APKMALDH1A1KMT2ANPSR1
SCHEMBL451772 0.82 SLC7A5 (0.62) SLC7A5PTPN1PTGS1PKMALPI
SCHEMBL4962288 0.82 RAB9A (0.50) RAB9ASLC7A5PTPN1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144388-A1 ACYL DERIVATIVES WHICH TREAT VLA-4 RELATED DISORDERS Elan Pharmaceuticals, Inc. (US) 2001-10-17 EP claimed
EP-1144384-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2001-10-17 EP claimed
WO-2000043372-A1 ACYL DERIVATIVES WHICH TREAT VLA-4 RELATED DISORDERS ELAN PHARMACEUTICALS, INC. (US) 2000-07-27 WO claimed
WO-2000043369-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2000-07-27 WO claimed
EP-1144384-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2001-10-17 EP disclosed
WO-2000043369-A1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2000-07-27 WO disclosed