SCHEMBL740058

SCHEMBL740058

COCCCn1c(C2CCCN(C(=O)CC(Cc3ccc4ccccc4c3)NC(=O)OC(C)(C)C)C2)nc2ccc(OC)nc21

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
PPIA P62937 2/20 0.35
PADI4 Q9UM07 2/20 0.34
KLK5 Q9Y337 1/20 0.34
GHSR Q92847 1/20 0.34
HRH1 P35367 3/20 0.33
KCNH2 Q12809 3/20 0.33
HRH2 P25021 1/20 0.33
MCHR1 Q99705 4/20 0.32
ACE P12821 1/20 0.32
TACR1 P25103 1/20 0.32
CYP2D6 P10635 2/20 0.32
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762621 1.00 CTSB (0.35) CTSBCTSSCTSKPPIAPADI4
SCHEMBL740059 1.00 CTSB (0.35) CTSBCTSSCTSKPPIAPADI4
SCHEMBL763177 0.93 CTSB (0.36) CTSBCTSSCTSKPPIAPADI4
SCHEMBL741997 0.92 KCNH2 (0.35) HRH1KCNH2MCHR1TACR1CYP2D6
SCHEMBL762559 0.89 KCNH2 (0.39) CTSBCTSSCTSKPADI4KLK5
SCHEMBL762785 0.89 HRH1 (0.42) CTSBCTSSCTSKPADI4HRH1
SCHEMBL762577 0.88 CTSB (0.36) CTSBCTSSCTSKPPIAPADI4
SCHEMBL762648 0.88 HRH1 (0.36) CTSBCTSSCTSKPPIAPADI4
SCHEMBL762513 0.87 KCNH2 (0.36) CTSBCTSSCTSKPADI4KLK5
SCHEMBL762657 0.87 PPARA (0.36) CTSBCTSSCTSKPPIAPADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed