SCHEMBL7400778

SCHEMBL7400778

CCOC=Cc1nc(N)nc(SCCc2ccccn2)c1C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
MAPT P10636 5/20 0.39
HPGD P15428 3/20 0.39
POLB P06746 1/20 0.39
PKM P14618 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ADORA1 P30542 5/20 0.38
ADORA3 P0DMS8 2/20 0.38
ADORA2A P29274 2/20 0.38
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HSD17B10 Q99714 3/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
SLC29A1 Q99808 3/20 0.35
GAA P10253 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441746 0.83 ALDH1A1 (0.48) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6441219 0.78 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6441876 0.78 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6441928 0.76 ADORA1 (0.46) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6441705 0.76 ADORA1 (0.59) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6440658 0.75 ADORA1 (0.44) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL7400049 0.75 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6444027 0.74 ADORA2A (0.54) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6443374 0.73 ADORA1 (0.55) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL6444649 0.73 ADORA2A (0.52) ALDH1A1MEN1KMT2AMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261327-A2 ADENOSINE RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2002-12-04 EP disclosed
WO-2001062233-A2 ADENOSINE RECEPTOR MODULATORS F. HOFFMANN LA ROCHE AG (CH) 2001-08-30 WO disclosed