SCHEMBL7401272

SCHEMBL7401272

O=C(O)CCNNC(=O)c1ccncc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.64
HDAC1 Q13547 1/20 0.64
HDAC2 Q92769 1/20 0.64
ALDH1A1 P00352 1/20 0.60
CYP1A2 P05177 2/20 0.58
CYP2C19 P33261 2/20 0.58
CYP2C9 P11712 1/20 0.58
KDM4E B2RXH2 1/20 0.52
MPO P05164 1/20 0.52
CYP3A4 P08684 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2A6 P11509 1/20 0.52
TP53 P04637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
GAA P10253 5/20 0.50
CA1 P00915 3/20 0.49
CA9 Q16790 3/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658753 0.84 CA12 (0.57) HDAC3HDAC1HDAC2GAACA1
SCHEMBL3203823 0.82 CYP1A2 (0.76) HDAC2ALDH1A1CYP1A2CYP2C19CYP2C9
Hydrochloric Acid SCHEMBL8658432 0.82 CA12 (0.56) HDAC3HDAC1HDAC2GAACA1
SCHEMBL2998085 0.82 ALDH1A1 (0.64) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL2998521 0.82 HDAC3 (0.68) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL3001447 0.81 HDAC3 (0.81) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL8248746 0.81 HTT (0.60) HDAC3HDAC1HDAC2ALDH1A1TDP1
Metazide SCHEMBL2109857 0.80 ALDH1A1 (0.72) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL9335619 0.79 MAPT (0.54) HDAC3HDAC1HDAC2ALDH1A1CYP2C19
SCHEMBL2994741 0.79 TDP1 (0.68) ALDH1A1CYP1A2CYP2C19CYP2C9TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255748-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-13 EP disclosed
WO-2001060813-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-23 WO disclosed