SCHEMBL7405141

SCHEMBL7405141

Oc1cc(C(F)(F)F)nn1-c1ccc(Cl)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.44
PTGS2 P35354 4/20 0.44
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ORAI1 Q96D31 1/20 0.38
CRACR2A Q9BSW2 3/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31199040 0.84 CRACR2A (0.42) CNR1CNR2CRACR2A
SCHEMBL31199062 0.84 MAPT (0.44) CNR1CNR2NPSR1CRACR2AKDM4E
SCHEMBL21919217 0.82 PTGS2 (0.42) PTGS1PTGS2CNR1CNR2
SCHEMBL18604839 0.81 KLKB1 (0.47) PTGS1PTGS2CNR1CNR2ORAI1
SCHEMBL31199164 0.80 EGLN2 (0.43) PTGS2CYP2C9CRACR2A
SCHEMBL7402120 0.78 PTGS2 (0.65) PTGS1PTGS2CYP1A2CYP3A4CYP2C9
SCHEMBL3106823 0.78 PTGS2 (0.46) PTGS1PTGS2CYP2C9
SCHEMBL6389262 0.78
SCHEMBL7407050 0.78 PTGS1 (0.39) PTGS1PTGS2CYP1A2CYP3A4CYP2C9
SCHEMBL31199118 0.77 UBE2T (0.44) CNR1CNR2CYP2C9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750550-A RESPIRATORY SYSTEM DISORDERS SANOFI (FR) 1998-05-12 US disclosed
WO-1997010243-A1 2-(PYRAZOL-5-YL-OXYMETHYL)-1,2-BENZISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (US) 1997-03-20 WO disclosed