SCHEMBL7405388

SCHEMBL7405388

O=C(O)C(CNC(=O)C1CC(CCCCNc2nc3c([nH]2)CCCC3)ON1)NS(=O)(=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.50
ITGAV P06756 13/20 0.50
ITGA2B P08514 10/20 0.50
ADAMTS4 O75173 1/20 0.39
MMP2 P08253 6/20 0.37
MMP9 P14780 5/20 0.37
MMP8 P22894 3/20 0.37
MMP12 P39900 3/20 0.37
MMP14 P50281 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401828 0.96 ITGB3 (0.48) ITGB3ITGAVITGA2B
SCHEMBL7408996 0.91 ITGB3 (0.52) ITGB3ITGAVITGA2B
SCHEMBL7406862 0.90 ITGB3 (0.53) ITGB3ITGAVITGA2B
SCHEMBL7403882 0.89 ITGB3 (0.53) ITGB3ITGAVITGA2B
SCHEMBL7399454 0.88 ITGB3 (0.51) ITGB3ITGAVITGA2B
SCHEMBL7404043 0.87 ITGB3 (0.52) ITGB3ITGAVITGA2BADAMTS4MMP2
SCHEMBL7400646 0.87 ITGB3 (0.53) ITGB3ITGAVITGA2BADAMTS4MMP2
SCHEMBL7399857 0.86 ITGB3 (0.50) ITGB3ITGAVITGA2B
SCHEMBL7405452 0.84 ITGB3 (0.53) ITGB3ITGAVITGA2BMMP2MMP9
SCHEMBL7403933 0.84 ITGB3 (0.70) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP claimed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO claimed
US-6214834-B1 ANGIOGENESIS INHIBITORS; ANTIINFLAMMATORY AGENTS; ANTICANCER AGENTS DUPONT PHARMACEUTICALS COMPANY 2001-04-10 US disclosed
WO-1996037492-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-11-28 WO disclosed