SCHEMBL7406235

SCHEMBL7406235

CCC(c1ccc(Cl)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.82

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 7/20 0.82
NQO1 P15559 5/20 0.72
VKORC1 Q9BQB6 3/20 0.62
KDM4E B2RXH2 1/20 0.62
ALDH1A1 P00352 1/20 0.62
ALB P02768 1/20 0.62
PCSK7 Q16549 1/20 0.62
HSD17B10 Q99714 1/20 0.62
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
CRHBP P24387 1/20 0.61
CASP7 P55210 1/20 0.61
CASP6 P55212 1/20 0.61
CRHR2 Q13324 1/20 0.61
HIF1A Q16665 1/20 0.61
TOP1 P11387 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenprocoumon SCHEMBL29392123 0.91 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL24500472 0.91 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL43031 0.91 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
Phenprocoumon SCHEMBL24500477 0.91 CYP2C9 (1.00) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7351110 0.90 CYP2C9 (0.87) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL7350773 0.87 CYP2C9 (0.82) CYP2C9NQO1VKORC1KDM4EALDH1A1
Coumachlor SCHEMBL30930052 0.86 CYP2C9 (0.84) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL1649090 0.86 CYP2C9 (0.73) CYP2C9NQO1VKORC1KDM4EALDH1A1
Coumachlor SCHEMBL433455 0.86 CYP2C9 (0.84) CYP2C9NQO1VKORC1KDM4EALDH1A1
SCHEMBL8042698 0.86 CYP2C9 (0.86) CYP2C9NQO1VKORC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed
US-4011332-A RODENTICIDE BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DT) 1977-03-08 US disclosed