SCHEMBL740778

SCHEMBL740778

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccccc4)cc3)NC(=O)O)C2)nc2cccc(Cl)c21

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMEL1 Q495T6 1/20 0.38
CYP2D6 P10635 4/20 0.37
HRH1 P35367 4/20 0.37
HSD11B1 P28845 4/20 0.37
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
KCNH2 Q12809 4/20 0.36
BTK Q06187 2/20 0.35
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
CHRM1 P11229 2/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739361 0.93 HRH1 (0.35) CYP2D6HRH1HSD11B1ALDH1A1TSHR
SCHEMBL762504 0.92 HRH1 (0.37) MMEL1CYP2D6HRH1ALDH1A1TSHR
SCHEMBL742063 0.92 KCNH2 (0.36) CYP2D6HRH1ALDH1A1TSHRLMNA
SCHEMBL740436 0.90 HRH1 (0.38) CYP2D6HRH1HSD11B1ALDH1A1TSHR
SCHEMBL740437 0.90 HRH1 (0.38) CYP2D6HRH1HSD11B1ALDH1A1TSHR
SCHEMBL740088 0.89 HRH1 (0.45) CYP2D6HRH1KCNH2CHRM1
SCHEMBL741369 0.89 MMEL1 (0.38) MMEL1CYP2D6HRH1HSD11B1ALDH1A1
SCHEMBL740692 0.86 HRH1 (0.35) CYP2D6HRH1HSD11B1ALDH1A1TSHR
SCHEMBL740312 0.86 HRH1 (0.45) CYP2D6HRH1KCNH2CHRM1
SCHEMBL739892 0.85 HRH1 (0.43) CYP2D6HRH1KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed